Description
Cyproterone is a steroidal anti-androgen that inhibits entry of androgens into the prostate. The acylated derivative of this compound is more potent and is used clinically more often.
Product Unit Size | Cost | Quantity | Stock |
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Cyproterone is a steroidal anti-androgen that inhibits entry of androgens into the prostate. The acylated derivative of this compound is more potent and is used clinically more often.
Cas No. | 427-51-0 |
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Purity | ≥98% |
Formula | C24H29ClO4 |
Formula Wt. | 416.94 |
Chemical Name | (1β,2β)-6-Chloro-1,2-dihydro-17-hydroxy-3'H- cyclopropa[1,2]pregna-1,4,6-triene-3,20-dione acetate |
IUPAC Name | [(1S,2S,3S,5R,11R,12S,15R,16S)-15-acetyl-9-chloro-2,16-dimethyl-6-oxo-15-pentacyclo[9.7.0.02,8.03,5.012,16]octadeca-7,9-dienyl] acetate |
Synonym | CPA, Androcur, Cyprostat |
Melting Point | 200-201°C |
Solubility | Soluble in dichloromethane and methyl alcohol. |
Appearance | White or almost white crystalline powder |
Store Temp | -20°C |
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Ship Temp | Ambient |
MSDS | |
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Info Sheet |
Guadalix FJ, Botella Llusiá J. The action mechanism of cyproterone. Acta Ginecol (Madr). 1975 Jul 1;27(1):7-11. PMID: 1146472.
Giorgi EP, Shirley IM, Grant JK, et al. Androgen dynamics in vitro in the human prostate gland. Effect of cyproterone and cyproterone acetate. Biochem J. 1973 Mar;132(3):465-74. PMID: 4125095.
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